Examples of 'agonist activity' in a sentence
Meaning of "agonist activity"
This phrase is used in the context of pharmacology or biology to describe the ability of a substance or drug to activate or stimulate certain receptors in the body. It refers to the degree or extent to which a substance can elicit a response or produce a specific biological effect
How to use "agonist activity" in a sentence
Basic
Advanced
agonist activity
These antibodies are devoid of any agonist activity.
Direct agonist activity has been demonstrated in two ways.
Some exhibit partial agonist activity.
Little agonist activity is shown.
The amount of label incorporated is indicative of agonist activity.
Agonist activity of antibody.
Antagonistic activity was not evaluated because of agonist activity.
Compounds to be tested for agonist activity were dissolved and diluted in buffer.
Those compounds are characterised as having benzodiazepine agonist activity.
Compounds of this class have some agonist activity at opioid receptors.
In preclinical studies enzalutamide lacks androgen receptor agonist activity.
Specific antibodies with agonist activity for the same receptors.
This activity has been termed inverse agonist activity.
Agonist activity was measured by the ability of the test compound to induce rotation.
This had the effect of reducing agonist activity.
See also
ND signifies that agonist activity was not detected.
Inhibition of cytokine release is indicative of the agonist activity.
The biologically active peptide exhibits agonist activity prior to insertion into the antibody framework.
These compounds are stated to have acetylcholine agonist activity.
Agonist activity was assessed by measuring changes in intracellular cyclic AMP.
The engineered antibodies of the invention exhibit agonist activity.
Compounds of the Invention having agonist activity may be either full or partial agonists.
This active principle is a GnRH hormone analogue with agonist activity.
Amino acids important for NPS agonist activity have been identified through Ala scanning mutagenesis.
This invention relates to muscarinic receptor ligands with agonist activity.
Measurement of agonist activity.
Assessment of these activities in response to a candidate compound is diagnostic of agonist activity.
This assay may be used to screen for agonist activity at this receptor.
Pharmacological activity may be assessed in functional in vitro assays of glucocorticoid agonist activity.
Aggregation at this point was indicative of agonist activity of the test compound.
This compound produced no PI turnover when administered by itself suggesting a lack of agonist activity.
None of these stereoisomers exhibit evidence of agonist activity in the in vitro functional assay.
The novel compounds of the present invention display melatonergic agonist activity.
This selectivity is demonstrated in the following agonist activity assays and receptor binding assays.
Antagonistic activity was not evaluated because the analogs possessed significant agonist activity.
To demonstrate AR agonist activity.
Their structures include a common vanilloid ring which appears to be important for agonist activity.
An antiarrhythmic effect, lack of partial agonist activity or intrinsic sympathomimetic activity.
Cells migrate across the permeable membrane towards compounds with agonist activity.
In vivo, they show an agonist activity at the level of these receptors.
The cycle is repeated until the desired affinity or agonist activity is achieved.
Agonist activity at the mu-receptor also causes suppression of opiate withdrawal.
Dye loaded cells were initially exposed to test compound to verify a lack of agonist activity.
In addition, agonist activity is enhanced relative to the straight chain derivatives.
Functional assay is used to differentiate between the agonist activity and the antagonist activity.
Polyamine-like agonist activity principally involves the carboxyl terminus.
Test compound was also evaluated alone at the indicated concentrations to test for agonist activity.
In the present invention, an agonist activity can be measured by a variety of assays.
This observed effect on plasma calcium is considered typical of amylin and calcitonin agonist activity.
Telmisartan does not exhibit any partial agonist activity at the AT1receptor.
You'll also be interested in:
Examples of using Agonist
Show more
The agonist and antagonist activities were measured
Varenicline is a partial agonist of the nicotine receptor
An agonist may function in a direct or indirect manner
Examples of using Activity
Show more
There is a lot of activity happening in that room
Activity cards divided into four themes
Refrain from physical activity until symptoms are gone
