Examples of 'competitive antagonist' in a sentence
Meaning of "competitive antagonist"
competitive antagonist: In pharmacology, a competitive antagonist is a type of receptor antagonist that binds to the receptor and blocks the physiological response, but unlike an irreversible antagonist, it can be displaced by increasing the concentration of the agonist
How to use "competitive antagonist" in a sentence
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competitive antagonist
It is also a competitive antagonist of the ionotropic glycine receptor.
This effect indicates that alcaftadine is a competitive antagonist of the receptor.
It acts as a competitive antagonist of the nicotinic acetylcholine receptor nAChR.
This value is considered to be a measure of the affinity of the competitive antagonist.
Caffeine is a competitive antagonist of GlyR.
By the selective abrogation of receptor subunit binding, a competitive antagonist is created.
Oxytocin which is a competitive antagonist of human oxytocin at receptor level.
The most frequently used drug is naltrexone, a long-acting competitive antagonist.
A competitive antagonist competes with an agonist for binding to the receptor.
Irreversible competitive antagonist.
A competitive antagonist is a receptor antagonist that binds to a receptor but fails to activate it.
Reversible competitive antagonist.
A competitive antagonist ( or competitive blocker ) competes with the neurotransmitter for the same binding site.
In doing this it is also acting as a competitive antagonist for the EGF ligand.
Naltrexone is a competitive antagonist for opioid receptors, effectively blocking the effects of endorphins and opioids.
See also
For example, the CGRP peptide antagonist can act as a competitive antagonist or a noncompetitive antagonist.
It is a competitive antagonist of aldosterone.
An example of such a peptide is a CD40 ligand competitive antagonist.
Naloxone is a pure competitive antagonist of opiate receptors and has no agonistic activity.
In some embodiments, the LFA-1 antagonist is a directly competitive antagonist.
It is a competitive antagonist.
This response was completely blocked by 20 µM capsazepine, a selective competitive antagonist of VR1.
Bicuculline is a competitive antagonist at the GABA binding site of GABAA receptors.
This variant, designated HGF/NK2, has been proposed to be a competitive antagonist of mature huHGF.
Icatibant was shown to be a competitive antagonist when the bradykinin challenge dose was increased 4-fold.
A competitive antagonist ( or competitive blocker ) interacts with or near the site specific for agonist binding.
These effects parallel that of AP-5, a competitive antagonist at NMDA receptors.
A competitive antagonist ( also known as a competitive blocker ) competes with an agonist for overlapping binding sites.
Identified antagonists include the competitive antagonist capsazepine and the non-competitive antagonist ruthenium red.
Naltrexoneis a competitive antagonist for opioid receptors, effectively blocking the effects of endorphins and opiates.
Atropine is a non-selective competitive antagonist with Acetylcholine at muscarinic receptors.
It 's a competitive antagonist of the A1 and A2a receptors of adenosine.
Iodoresiniferatoxin ( I-RTX ) is a strong competitive antagonist of the Transient Receptor Potential Vanilloid 1 ( TRPV1 ) receptor.
Naloxone is a competitive antagonist and large doses ( 4 mg ) may be required in seriously poisoned patients.
Icatibant is a selective competitive antagonist of BK2R and ecallantide inhibits the action of kallikrein.
It is a weak competitive antagonist of the androgen receptor ( AR ) and a potent 5α-reductase inhibitor.
Icatibant is a selective competitive antagonist at the bradykinin type 2 ( B2 ) receptor.
It is a weak competitive antagonist of the androgen receptor (AR).
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Examples of using Competitive
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They get really competitive about it too
Competitive in terms of both price and technology
Your mistake was getting competitive with a machine
Examples of using Antagonist
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You are the final antagonist in the game
Antagonist drugs could provide better recover
Who is the principal antagonist in the strike
