Examples of 'full agonist' in a sentence
Meaning of "full agonist"
full agonist: In pharmacology, a 'full agonist' refers to a substance that binds to and activates a receptor in the body to produce a maximum response
How to use "full agonist" in a sentence
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full agonist
Mexamine is a full agonist to several serotonin receptors.
The response is measured relative to a full agonist like dopamine.
It is a full agonist of the benzodiazepine receptor.
Buprenorphine has a low abuse liability compared to full agonist opioids.
The agonist includes a full agonist and a partial agonist.
Full agonist is a substance that produces a full response or the maximum effect at a given receptor.
Sufentanil acts as a full agonist in µ-opioid receptors.
Full agonist opioids activate the opioid receptors fully resulting in the full opioid effect.
Sufentanil acts as a full agonist in μ-opioid receptors.
However, antagonists cause no opioid effect and block full agonist opioids.
Existing full agonist compounds such as terlipressin have a narrow therapeutic index.
Perform antagonist dose responses in the presence of a saturating dose of full agonist ( methanandamide ).
It is a highly discerning full agonist that possesses a highly affinity for the prostaglandin FP receptor.
Cross-tolerance has also been shown between bretazenil and full agonist benzodiazepines in rats.
Thus, a compound may be a full agonist in a given tissue but a partial in others.
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Higher activity numbers indicate higher efficacy relative to carbachol, a full agonist at all muscarinic receptors.
It acts as a full agonist at cannabinoid receptors type 1 and 2.
In some embodiments, the PPAR gamma modulator is a full agonist or a partial agonist.
It behaves as a full agonist at the D1 protomer and a high-affinity partial agonist at the D2 protomer.
In a further embodiment said peptide is a full agonist of the melanocortin receptor MC1 r.
A full agonist at the 5-HT1D receptor is most preferred.
A model of PPAR activation by a full agonist and a partial agonist is given in Fig . 1.
A full agonist at the 5-HT1A receptor is most preferred.
In a further case said peptide is a full agonist of the melanocortin receptor MC1 r.
A full agonist at the the 5-HT1B receptor is most preferred.
Figure 1 illustrates a model of PPAR activation by a full agonist and a partial agonist, respectively.
Norepinephrine is the standard full agonist used for evaluating alpha-1 and alpha-2 receptor activity.
Doxanthrine is a synthetic compound which is a potent and selective full agonist for the dopamine D1 receptor.
For these experiments, the full agonist is defined as Norepinephrine ( NE ) bitartrate ( control ).
As used herein, " modulator " means both antagonist, partial or full agonist and inverse agonist.
The term " agonist " means full agonist or partial agonist.
It acts as a potent and selective 5-HT1A receptor full agonist.
Studies have shown that strontium is a full agonist of the calclum-sensing receptor ( CaR ).
The m5D5 was used as a dose-dependent full agonist control.
Nevertheless Compound 16 is a full agonist to cause coronary vasodilation.
However, only the heterodimer ( A ), not the homodimer ( B ) acts as a full agonist to induce signaling.
In the acetic acid writhing assay, 6d displayed full agonist activity with a calculated A50 value of 7.5 nmol.
Results are presented normalized to the full agonist N-6-cyclopentyladenosine, CPA.
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Examples of using Agonist
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The agonist and antagonist activities were measured
Varenicline is a partial agonist of the nicotine receptor
An agonist may function in a direct or indirect manner
Examples of using Full
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The world was full of startling new concepts
Full transition to new system of administration of justice
They are always full of coy little tricks
