Examples of 'receptor affinity' in a sentence
Meaning of "receptor affinity"
Receptor affinity: The strength of the interaction between a receptor and a ligand, often used in pharmacology to describe how well a drug binds to its target receptor
How to use "receptor affinity" in a sentence
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receptor affinity
Insulin receptor affinity relative to human insulin.
Saturation binding analysis can determine receptor affinity and density.
Receptor affinity can be measured using standard methodology such as is described below.
The drug does not appear to affect receptor affinity for gonadotropins.
The receptor affinity of candidate compounds can be determined by radioligand binding competition studies.
The thesis developed the concepts of receptor affinity and intrinsic activity.
The method was used to monitor the effects of conjugation and oxidation on receptor affinity.
The insulin receptor affinity of the compounds of this invention are within the desired range.
Another aspect relates to the furnishing of insulin derivatives having a low insulin receptor affinity.
The desired dose depends on its receptor affinity and availability at the receptor site.
The truncated molecule exhibits reduced biological activity while maintaining high receptor affinity.
Immobilized eck - x receptor affinity chromatography.
Supplementing the parenteral infusate with exogenous GIP resulted in a further reduction in insulin receptor affinity.
Thus, concerns about receptor affinity states are eliminated.
As a result, the compounds of the present invention exhibited good NMDA receptor affinity.
See also
A parallel reduction in? - adrenergic receptor affinity for agonists was also seen.
Certain compounds of Formula ( I ) exhibit increased delta opioid receptor affinity.
Preferably, the adhesins are purified by receptor affinity chromatography or monoclonal antibody affinity chromatography.
All compounds of Examples showed selective CB2 receptor affinity.
Table 4 provides glucagon receptor affinity and antagonist activity for several specific glucagon analog antagonists.
Preferably, the protein is further purified by receptor affinity chromatography.
Muscarinic receptor affinity test ( in vitro ).
As mentioned above, suitable CRF antagonists include compounds which demonstrate CRF receptor affinity.
The results of compounds with a good hNK-3 receptor affinity are shown in the following Table 1.
A structurally novel class of compounds has now been found which also possess 5-HT6 receptor affinity.
Receptor affinity profiles in radioligand binding assays Receptor Affinity [ k1 ( nM ) ].
The EC50 is calculated as a measure of receptor affinity.
Example 178, Insulin receptor affinity of selected insulin derivatives of the invention,.
All of the AIB-containing peptides have higher ORL-1 receptor affinity than the native NC ligand.
The 5-HT2A receptor affinity values are expressed as Ki values.
All compounds of Examples showed 5HT4 receptor affinity.
However, this structural modification resulted in a 67-fold decrease in CB1 receptor affinity.
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Examples of using Affinity
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Expose his unholy affinity for savages
My affinity with the radio operator was confirmed
We have a basic affinity for our family
Examples of using Receptor
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Receptor is not sensitive to the type of change
Is that why that receptor network existed
This receptor can exist in three conformations
