Examples of 'receptor antagonist activity' in a sentence
Meaning of "receptor antagonist activity"
Receptor antagonist activity: In pharmacology and biology, this phrase pertains to the ability of a substance to block or inhibit the action of specific receptors in the body. Antagonists bind to receptors without activating them, thereby producing a physiological response that is different from that of agonists
How to use "receptor antagonist activity" in a sentence
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receptor antagonist activity
Compounds of this invention possess muscarinic receptor antagonist activity.
NK3 receptor antagonist activity was determined for a subset of the 17 compounds.
Buspirone expresses both serotonin and dopamine receptor antagonist activity.
A particular compound possessing endothelin receptor antagonist activity is YM598 or a pharmaceutically acceptable salt thereof.
Any molecule or compound can be screened for chemokine receptor antagonist activity.
A particular compound possessing endothelin receptor antagonist activity is ZD1611 or a pharmaceutically acceptable salt thereof.
The compounds of the invention have excellent mineralocorticoid receptor antagonist activity.
This compound has 5-HT4 receptor antagonist activity.
The present invention relates to a series of new heterocyclic compounds having tachykinin receptor antagonist activity.
Inhibition of contraction demonstrates angiotensin II receptor antagonist activity of the test compound.
Intermediates for use in the preparation of urea compounds having muscarinic receptor antagonist activity.
Representative compounds are tested for 5-HT1A receptor antagonist activity in the cAMP assay.
The indanyl compounds of the invention are compounds having a calcium receptor antagonist activity.
These compounds have 5-HT4 receptor antagonist activity.
Rupatadine is a second generation, non-sedating, long-acting histamine antagonist with selective peripheral H1 receptor antagonist activity.
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These metabolites possess minimal NMDA receptor antagonist activity.
The invention provides novel compounds that possess mu opioid receptor antagonist activity.
These metabolites have minimal NMDA receptor antagonist activity.
Compounds of this invention possess both B2 adrenergic receptor agonist activity and muscarinic receptor antagonist activity.
Heterocycle derivative having pgd2 receptor antagonist activity.
Fexofenadine is a well-known antihistamine compound which has a selective peripheral H1 receptor antagonist activity.
These compounds have H3 histamine receptor antagonist activity.
In some embodiments, the compounds provided herein exhibit tissue selective androgen receptor antagonist activity.
These metabolites each have less than 1 % of the 5-HT3 receptor antagonist activity of palonosetron.
Refers to certain heterocyclic carboxamide derivatives which are disclosed as having 5-HT4 receptor antagonist activity.
This in vivo activity appears to be the result of NMDA receptor antagonist activity.
Desloratadine is a non-sedating, long-acting histamine antagonist with selective peripheral H1 - receptor antagonist activity.
Compounds of formula I possess muscarinic receptor antagonist activity.
The extracts obtained from this novel strain have a very advantageous NPY receptor antagonist activity.
The compound of formula I has muscarinic receptor antagonist activity.
Biphenyl derivatives having b sb 2 / sb adrenergic receptor agonist and muscarinic receptor antagonist activity.
These compounds are stated to exhibit serotonin M receptor antagonist activity.
This selectivity is demonstrated in the following receptor binding assays and receptor antagonist activity assays.
Numerous chemical substances are known to have histamine-H, receptor antagonist activity.
Preferably, the peptide of and for use in the invention has bradykinin B2 receptor antagonist activity.
The compounds are additionally disclosed to have H1 receptor antagonist activity.
Numerous chemical substances are known to have histamine H1 receptor antagonist activity.
In particular, Pharmaceutical Compounds exhibit metabotropic glutamate receptor antagonist activity.
Lastly, a protein inhibitor, purified and cloned, that has interleukin-1 receptor antagonist activity has been reported.
These compounds exhibit dopamine antagonist and 5-HT ₃ receptor antagonist activity.
Describes indole derivatives having 5-HT3 receptor antagonist activity.
UTILITY Compounds of the invention possess angiotensin II type 1 ( AT1 ) receptor antagonist activity.
Thus, many adenosine A1 receptor antagonists also possess some degree of A2 receptor antagonist activity.
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Examples of using Antagonist
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