Examples of 'partial agonist' in a sentence
Meaning of "partial agonist"
partial agonist - A partial agonist is a type of drug or substance that binds to and activates a specific receptor in the body but produces a smaller or more moderate response compared to a full agonist. This term is commonly used in pharmacology and medicine to describe the partial efficacy of certain medications.
How to use "partial agonist" in a sentence
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partial agonist
Varenicline is a partial agonist of the nicotine receptor.
It was concluded that it may be an opioid partial agonist.
The partial agonist is therefore acting as an antagonist.
The agonist may be a partial agonist.
It is a partial agonist at some opioid receptors and an antagonist at another.
An agonist may be a full or partial agonist.
These tests may suggest partial agonist or a functional antagonist activity.
The agonist includes a full agonist and a partial agonist.
Some exhibit partial agonist activity.
A partial agonist produces only a partial physiological response of the endogenous ligand.
Very weak partial agonist.
Partial agonist are often difficult to differentiate from full agonists in functional assays.
This profile of action may reflect partial agonist properties.
A receptor partial agonist is a substance which binds receptor and partially activate them.
A selective androgen receptor agonist or partial agonist may be used as an anabolic agent.
See also
Cariprazine has partial agonist as well as antagonist properties depending on the endogenous dopamine levels.
It might be argued that the endogenous agonist is simply a partial agonist in that tissue.
It is a partial agonist for GABAA receptors in the brain.
An agonist that can only partially activate the physiological response is called a partial agonist.
Here it acts as a low affinity partial agonist of the benzodiazepine receptor.
A partial agonist partially opens the NMDA receptor channel.
Acts as a partial agonist.
Buprenorphine is not a silent antagonist of the KOR but rather a weak partial agonist.
Buprenorphine is a synthetic opioid partial agonist with mixed agonist and antagonist properties.
The reduction in the NGF neurotrophic response correspond to a profile of a partial agonist of NGF.
A selective androgen receptor agonist or partial agonist is used for male hormone replacement therapy.
This is the first observation that a small moleucle BDNF mimetic can function as a partial agonist.
ACC is also an exogenous partial agonist of the mammalian NMDA receptor.
Certain embodiments provide a selective HGF partial agonist.
An antiarrhythmic effect, lack of partial agonist activity or intrinsic sympathomimetic activity.
It is a 3rd generation adrenergic β receptor partial agonist.
Telmisartan does not exhibit any partial agonist activity at the AT1receptor.
In one embodiment, the modulating antibody is a positive modulator or partial agonist.
Due to partial agonist characteristic, has limited addictive and respiratory depressant properties.
In some embodiments, the agonist is a partial agonist.
Indacaterol is a partial agonist at the human beta2-adrenergic receptor with nanomolar potency.
Alternatively, the antagonist can be a partial agonist.
In vivo, they show an agonist or partial agonist activity with respect to these receptors.
In one approach, the modulating antibody is a positive modulator or partial agonist.
More specifically, partial agonist activity can be measured according to the following procedures.
The present invention may act as an agonist, partial agonist or antagonist.
Buprenorphine is a partial agonist at the µ-opioid receptor and an antagonist at the k-opioid receptor.
In another embodiment the compound is an inverse agonist, partial agonist or partial antagonist.
Further, the partial agonist properties of buprenorphine are useful in the treatment of opioid addiction.
In certain embodiments, the method comprises identifying a partial agonist of the receptor.
Buprenorphine is a partial agonist at the mu-opiate receptor and chronic administration can produce opioid dependence.
In yet other embodiments, the compound may be a partial agonist of said receptor.
A 5HT1A partial agonist known as buspirone is currently being marketed as an anxiolytic agent.
The method of claim 2 wherein the directly identified compound is a partial agonist.
A selective androgen receptor agonist and / or partial agonist may be used to improve athletic performance.
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Examples of using Agonist
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The agonist and antagonist activities were measured
Varenicline is a partial agonist of the nicotine receptor
An agonist may function in a direct or indirect manner
Examples of using Partial
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Partial allowance for special dangerous goods
They even found a partial on the handcuffs
Partial inspections are done on each shutdown if time allows
