Examples of 'partial agonists' in a sentence
Meaning of "partial agonists"
partial agonists: In pharmacology, this term refers to drugs that bind to and activate a specific type of receptor in the body, producing a partial physiological response
How to use "partial agonists" in a sentence
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partial agonists
There are several different types of partial agonists.
Partial agonists and receptor reserve.
This dual behavior is typical of partial agonists.
Partial agonists may be viewed from biochemical or physiological viewpoint.
This basically means that they are partial agonists.
The term includes partial agonists and inverse agonists.
Such behavior is characteristic of partial agonists.
Compounds considered partial agonists tend to have efficacy in between this range.
They are actually called partial agonists.
Partial agonists may activate the receptor less compared to isovaleric acid.
This is in particular the case for PPARdelta partial agonists.
They behave in vivo as complete or partial agonists with respect to these receptors.
Divalent antibodies of the prior art are agonists or partial agonists.
Partial agonists and full agonists are envisaged but full agonists are preferred.
This is in particular the case for PPARgamma partial agonists.
See also
Inverse agonists and partial agonists may under certain assay conditions be antagonists.
Certain of the compounds are also useful as glycine partial agonists.
Partial agonists may activate the receptor less compared to the carboxylic acid.
Certains of the compounds are also useful as glycine partial agonists.
The compounds of Formula I act as partial agonists on the dopamine receptors.
Agents that are only partly as effective as agonists are termed partial agonists.
In one aspect they are agonists or partial agonists of the relevant PPAR.
Compounds of the Invention having agonist activity may be either full or partial agonists.
The compounds of Formula I act as partial agonists on the monoaminergic neurotransmitter receptors.
The compounds as described herein may be glycine site NMDA receptor partial agonists.
Serotonin 7 partial agonists are useful for the treatment of depression.
FXR agonist may act as agonists or partial agonists of FXR.
Serotonin 7 partial agonists are also useful for the treatment of anxiety.
Compounds that reduce the transactivation by Avandia are PPAR partial agonists.
As such, agonists include partial agonists and full agonists.
Known subfunctionalities are full agonists, or partial agonists.
However, the mutants behaved as partial agonists in the proliferation assay.
Opioids are classified as agonists, antagonists and partial agonists.
In some embodiments, the compounds are partial agonists or partial antagonists in a tissue selective manner.
These long-acting metabolites are partial agonists.
Partial agonists and partial antagonists are also known and are encompassed by the term “ opioid ”.
This includes agonists, antagonists and partial agonists.
Partial agonists can also function as " blockers " by preventing the binding of more robust agonists.
The compounds are said to be agonists, partial agonists or antagonists in vivo.
Second, in the absence of polyamines, the derivatives can be viewed as partial agonists.
The compounds of the invention are partial agonists or antagonist at the dopamine D4 receptors.
The term agonists as used herein, includes partial agonists.
The compounds of the invention are partial agonists or antagonist at the dopamine D4 receptor.
In the present specification, the agonist includes full agonists and partial agonists.
Various agonists or partial agonists of B2 adrenergic receptors are known.
These compounds are disclosed as being serotonin agonists, partial agonists or antagonists.
Partial agonists are hence herein encompassed within the term " antagonist ".
The activating compounds can in particular be agonist compounds, partial agonists or positive allosteric modulators.
Partial agonists show a dualistic effect, i.e. they comprise agonistic as well as antagonistic effects.
Examples of ligands activating peroxisome proliferator-activated receptor gamma as partial agonists are honokiol and falcarindiol.
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